technetium tc-99m pyro/trimeta phosphates kit

Small moleculeapprovedImaging agent

Approved

Nov 19, 1976

Mebrofenin is a chelating component which, when attached to Technetium TC-99M, forms a diagnostic drug marketed under the name Choletec. Choletec is approved by FDA as a hepatobiliary imaging agent. — NCATS

Clinical trial activity

0 trials · 0 clinical orgs · 1 marketing orgs

Phase 1
0
Phase 2
0
Phase 3
0
Phase 4
0

Timeline

1970s

  1. Nov 19, 1976

    Pharmalucence — Earliest FDA Approval

  2. Nov 19, 1976

    Pharmalucence — NDA Secondary Org

  3. Nov 19, 1976

    Pharmalucence — NDA Organization

Indications

Mechanism of action

  • Unspecified targetRadiopharmaceutical

    Radiopharmaceutical

Approval history

  • approvedNov 19, 1976

Chemistry & pharmacology

Loading structure…

SMILES

[99Tc]
Mol. weight
98.91 g/mol
Chirality
Single Stereoisomer
Inorganic
No
Polymer
No
Delivery
Parenteral
Availability
Discontinued
Imaging
99-technetium

Oral

No

Parenteral

Yes

Topical

No

Sources

Also known as

  • pyrolite
  • pyrolite
  • technetium tc 99m (pyro- and trimeta-) phosphates
  • technetium tc-99m pyro/trimeta phosphates kit
  • technetium tc-99m pyro/trimeta phosphates kit
  • technetium tc-99m pyro/trimeta phosphates kit

Organizations

Marketing (2)

OrganizationOrg typeRelationshipDate
PharmalucenceFor profitNDA2Nov 19, 1976
PharmalucenceFor profitNDANov 19, 1976