phenindamine
Small moleculeexperimental
Phenindamine (thephorin or 2-methyl-9-phenyl-2,3,4,9-tetrahydro-1-pyridindene) a pyridindene derivative proved to be a potent antihistaminic. Phenindamine was used to treat sneezing; runny nose; itching, watery eyes; hives; rashes; itching; and other symptoms of allergies and the common cold. — NCATS
Clinical trial activity
0 trials · 0 clinical orgs · 0 marketing orgs
Phase 1
0
Phase 2
0
Phase 3
0
Phase 4
0
Indications
Approved for
Mechanism of action
- Histamine H1 receptorANTAGONIST
Histamine H1 receptor antagonist
Chemistry & pharmacology
Loading structure…
SMILES
CN1CCC2=C(C1)C(c1ccccc1)c1ccccc12- Mol. weight
- 261.37 g/mol
- Lipinski Ro5
- Pass
- Rule of 3
- No
- Chirality
- Racemic Mixture
- Inorganic
- No
- Polymer
- No
Oral
No
Parenteral
No
Topical
No
Sources
- ChEMBLCHEMBL278398 ↗
- WikipediaPhenindamine ↗
- NCATS772BQ8KSST ↗
- ChEMBLCHEMBL2107213 ↗
Also known as
- 2,3,4,9-tetrahydro-2-methyl-9-phenyl-lh-indeno- (2,1-c)pyridine
- allphar brand of phenindamine tartrate
- carnrick brand of phenindamine tartrate
- fenindamina
- fenindamina
- nolahist
- nolahist
- nolahist
- phenindamine
- phenindamine
- phenindamine
- phenindamine
- phenindamine
- phenindamine
- phenindamine
- phenindamine
- phenindamine hydrochloride
- phenindamine tartrate
- phenindamine tartrate
- phenindamine tartrate
- phenindamine tartrate
- phenindaminum
- phenindaminum
- phenindiamine
- phenindiamine
- theforin
- thephorin
- thephorin
- thephorin
- thephorin
- thephorin