rebaudioside

Small moleculeexperimental

Rebaudioside A is a steviol glycoside from the leaves of Stevia rebaudiana that is 240 times sweeter than sugar. Rebaudioside A is the sweetest and most stable steviol glycoside, and is less bitter than stevioside. Stevia leaves contain 9.1% stevioside and 3.8% rebaudioside A. — Wikipedia

Clinical trial activity

6 trials · 10 clinical orgs · 0 marketing orgs

Phase 1
3
Phase 2
1
Phase 3
0
Phase 4
0

Earliest trial started May 1, 2011 (NCT01403233)

Timeline

2010s

  1. Jan 1, 2011

    Earliest Phase 1 Sponsor(trial)

  2. Jan 1, 2012

    Earliest Phase 2 Sponsor(trial)

Indications

Mechanism of action

  • Unspecified target

    sweetener

Chemistry & pharmacology

Loading structure…

SMILES

C=C1C[C@@]23CC[C@H]4[C@@](C)(CCC[C@@]4(C)C(=O)O[C@@H]4O[C@H](CO)[C@@H](O)[C@H](O)[C@H]4O)[C@@H]2CC[C@]1(O[C@@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O[C@@H]1O[C@H](CO)[C@@H](O)[C@H](O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)[C@H]1O)C3
Mol. weight
967.02 g/mol
Lipinski Ro5
3 violation(s)
Rule of 3
No
Chirality
Single Stereoisomer
Inorganic
No
Polymer
No

Oral

No

Parenteral

No

Topical

No

Sources

Also known as

  • rebaudioside
  • rebaudioside
  • rebaudioside-a 303.7mg/day

Clinical trials

NCT IDPhaseStart dateSponsor(s)
NCT07018921N/AMar 15, 2023University of Manchester
NCT05287906N/AApr 15, 2022Cargill, MB Clinical Research and Consulting LLC, Midwest Center for Metabolic and Cardiovascular Research
NCT04991714Early Phase 1 (Phase 1)Aug 5, 2021University of Vienna
NCT03510624Phase 1Jun 1, 2018Katholieke Universiteit Leuven
NCT01757990Phase 2Mar 1, 2012University of Milan, University of Sassari
NCT01403233Phase 1May 1, 2011DSM, KGK Science Inc.
Showing 6 of 6 trials
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Organizations

Research & Development (10)

OrganizationOrg typeTrialsAs lead sponsorPhasesEarliest year
CargillFor profit1012022
DSMFor profit1112011
Katholieke Universiteit LeuvenAcademic/Hospital1112018
KGK Science Inc.For profit1012011
MB Clinical Research and Consulting LLCFor profit1012022
Midwest Center for Metabolic and Cardiovascular ResearchAcademic/Hospital1112022
University of ManchesterAcademic/Hospital1112023
University of MilanAcademic/Hospital1012012
University of SassariAcademic/Hospital1112012
University of ViennaAcademic/Hospital1112021
10 organizations
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