← Mechanisms of action

NOS1

SINGLE PROTEINHomo sapiens
Preferred name: Nitric-oxide synthase, brain ChEMBL ↗

Linked proteins

Drugs acting on this target (13)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
bz371aActivatorexperimentalSmall moleculeNOS1 activator
bz371bActivatorexperimentalPeptideNOS1 activator
yhd1023ActivatorexperimentalSmall moleculeNOS1 activator
gw 274150InhibitorexperimentalSmall moleculeNOS1 inhibitor
kd7040InhibitorexperimentalSmall moleculeNOS1 inhibitor
l-nmmaInhibitorexperimentalSmall moleculeNOS1 inhibitor
n-omega-nitro-l-arginine methyl esterInhibitorexperimentalSmall moleculeNOS1 inhibitor
nox-100InhibitorexperimentalSmall moleculeNOS1 inhibitor
nrgInhibitorexperimentalSmall moleculeNOS1 inhibitor
nxn-188InhibitorexperimentalSmall moleculeNOS1 inhibitor
nxn-462InhibitorexperimentalSmall moleculeNOS1 inhibitor
ronopterinInhibitorexperimentalSmall moleculeNOS1 inhibitor
tilarginineInhibitorexperimentalSmall moleculeNOS1 inhibitor