← Mechanisms of action
HTR1D
SINGLE PROTEINHomo sapiens
Preferred name: Serotonin 1d (5-HT1d) receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (12)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| almotriptan (axert) | Agonist | approved | Small molecule | HTR1D agonist |
| dihydroergotamine (D.H.E. 45) | Agonist | approved | Small molecule | HTR1D agonist |
| donitriptan | Agonist | experimental | Small molecule | HTR1D agonist |
| eletriptan (relpax) | Agonist | approved | Small molecule | HTR1D agonist |
| ergotamine | Agonist | approved | Small molecule | HTR1D agonist |
| fenfluramine (Pondimin) | Agonist | approved | Small molecule | HTR1D agonist |
| frovatriptan (frova) | Agonist | approved | Small molecule | HTR1D agonist |
| naratriptan (amerge) | Agonist | approved | Small molecule | HTR1D agonist |
| rizatriptan (maxalt) | Agonist | approved | Small molecule | HTR1D agonist |
| sumatriptan (zecuity) | Agonist | approved | Small molecule | HTR1D agonist |
| zolmitriptan (zomig) | Agonist | approved | Small molecule | HTR1D agonist |
| gsk163090 | Antagonist | experimental | Small molecule | HTR1D antagonist |