← Mechanisms of action
Bacterial DNA-directed RNA polymerase
PROTEIN COMPLEXBacteria
Linked proteins
Drugs acting on this target (6)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| rifamycin (aemcolo) | Antagonist | approved | Small molecule | Bacterial DNA-directed RNA polymerase antagonist |
| morinidazole | Inhibitor | experimental | Small molecule | Bacterial DNA-directed RNA polymerase inhibitor |
| rifabutin (mycobutin) | Inhibitor | approved | Small molecule | Bacterial DNA-directed RNA polymerase inhibitor |
| rifampin | Inhibitor | approved | Small molecule | Bacterial DNA-directed RNA polymerase inhibitor |
| rifapentine (priftin) | Inhibitor | approved | Small molecule | Bacterial DNA-directed RNA polymerase inhibitor |
| rifaximin (xifaxan) | Inhibitor | approved | Small molecule | Bacterial DNA-directed RNA polymerase inhibitor |