← Mechanisms of action
HRH2
SINGLE PROTEINHomo sapiens
Preferred name: Histamine H2 receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (11)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| betazole (histalog) | Agonist | approved | Small molecule | HRH2 agonist |
| cimetidine (tagamet) | Antagonist | approved | Small molecule | HRH2 antagonist |
| ebrotidine | Antagonist | experimental | Small molecule | HRH2 antagonist |
| famotidine (pepcid) | Antagonist | approved | Small molecule | HRH2 antagonist |
| methantheline bromide (banthine) | Antagonist | approved | Small molecule | HRH2 antagonist |
| nizatidine (axid) | Antagonist | approved | Small molecule | HRH2 antagonist |
| protecadin | Antagonist | experimental | Small molecule | HRH2 antagonist |
| ranitidine (zantac) | Antagonist | approved | Small molecule | HRH2 antagonist |
| lavoltidine | Inhibitor | experimental | Small molecule | HRH2 inhibitor |
| raluridine | Inhibitor | experimental | Small molecule | HRH2 inhibitor |
| rezatomidine | Inhibitor | experimental | Small molecule | HRH2 inhibitor |