← Mechanisms of action
EZH1
SINGLE PROTEINHomo sapiens
Preferred name: Histone-lysine N-methyltransferase EZH1 ChEMBL ↗
Linked proteins
Drugs acting on this target (4)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| gcb-002 | Inhibitor | experimental | Small molecule | EZH1 inhibitor |
| hh2853 | Inhibitor | experimental | Small molecule | EZH1 inhibitor |
| hm97662 | Inhibitor | experimental | Small molecule | EZH1 inhibitor |
| valemetostat (Ezharmia) | Inhibitor | experimental | Small molecule | EZH1 inhibitor |