← Mechanisms of action
RAF1
SINGLE PROTEINHomo sapiens
Preferred name: Serine/threonine-protein kinase RAF ChEMBL ↗
Linked proteins
Drugs acting on this target (18)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| lerafaon | Antisense inhibitor | experimental | Nucleic acid | RAF1 antisense inhibitor |
| arq 736 | Inhibitor | experimental | Small molecule | RAF1 inhibitor |
| cct3833 | Inhibitor | experimental | Small molecule | RAF1 inhibitor |
| gw5074 | Inhibitor | experimental | Small molecule | RAF1 inhibitor |
| isis 5132 | Inhibitor | experimental | Nucleic acid | RAF1 inhibitor |
| jzp815 | Inhibitor | experimental | Small molecule | RAF1 inhibitor |
| ly3009120 | Inhibitor | experimental | Small molecule | RAF1 inhibitor |
| nvp-lgx806 | Inhibitor | experimental | Small molecule | RAF1 inhibitor |
| plx-5568 | Inhibitor | experimental | Small molecule | RAF1 inhibitor |
| qlh11906 | Inhibitor | experimental | Small molecule | RAF1 inhibitor |
| regorafenib (stivarga) | Inhibitor | approved | Small molecule | RAF1 inhibitor |
| sorafenib (nexavar) | Inhibitor | approved | Small molecule | RAF1 inhibitor |
| spyk04 | Inhibitor | experimental | Small molecule | RAF1 inhibitor |
| tak-583 | Inhibitor | experimental | Small molecule | RAF1 inhibitor |
| tr128 | Inhibitor | experimental | Small molecule | RAF1 inhibitor |
| tr64 | Inhibitor | experimental | Small molecule | RAF1 inhibitor |
| vs-6766 | Inhibitor | experimental | Small molecule | RAF1 inhibitor |
| xl281 | Inhibitor | experimental | Small molecule | RAF1 inhibitor |