← Mechanisms of action
CNR1
SINGLE PROTEINHomo sapiens
Preferred name: Cannabinoid CB1 receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (35)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| acetaminophen (tylenol) | Agonist | approved | Small molecule | CNR1 agonist |
| beta-caryophyllene | Agonist | experimental | Small molecule | CNR1 agonist |
| jw0108 | Agonist | experimental | Small molecule | CNR1 agonist |
| jwh018 | Agonist | experimental | Small molecule | CNR1 agonist |
| nabilone (cesamet) | Agonist | approved | Small molecule | CNR1 agonist |
| Nabiximols | Agonist | experimental | Small molecule | CNR1 agonist |
| nonabine | Agonist | experimental | Small molecule | CNR1 agonist |
| org 28611 | Agonist | experimental | Small molecule | CNR1 agonist |
| sad-448 | Agonist | experimental | Small molecule | CNR1 agonist |
| aef0217 | Antagonist | experimental | Small molecule | CNR1 antagonist |
| ave-1625 | Antagonist | experimental | Small molecule | CNR1 antagonist |
| azd-2207 | Antagonist | experimental | Small molecule | CNR1 antagonist |
| cannabigerol | Antagonist | experimental | Small molecule | CNR1 antagonist |
| cp-741,952 | Antagonist | experimental | Small molecule | CNR1 antagonist |
| ibipinabant | Antagonist | experimental | Small molecule | CNR1 antagonist |
| oleoylethanolamide | Antagonist | experimental | Small molecule | CNR1 antagonist |
| otenabant | Antagonist | experimental | Small molecule | CNR1 antagonist |
| rimonabant | Antagonist | experimental | Small molecule | CNR1 antagonist |
| slv341 | Antagonist | experimental | Small molecule | CNR1 antagonist |
| surinabant | Antagonist | experimental | Small molecule | CNR1 antagonist |
| v24343 | Antagonist | experimental | Small molecule | CNR1 antagonist |
| aef0117 | Inhibitor | experimental | Small molecule | CNR1 inhibitor |
| pregnenolone | Inhibitor | experimental | Small molecule | CNR1 inhibitor |
| ryi-018 | Inhibitor | experimental | mAb | CNR1 inhibitor |
| syt-510 | Inhibitor | experimental | Small molecule | CNR1 inhibitor |
| crb-913 | Inverse agonist | experimental | Small molecule | CNR1 inverse agonist |
| gfb-024 | Inverse agonist | experimental | Small molecule | CNR1 inverse agonist |
| inv-101 | Inverse agonist | experimental | Small molecule | CNR1 inverse agonist |
| inv-202 | Inverse agonist | experimental | Small molecule | CNR1 inverse agonist |
| inv-347 | Inverse agonist | experimental | Small molecule | CNR1 inverse agonist |
| mk-9470 | Inverse agonist | experimental | Small molecule | CNR1 inverse agonist |
| taranabant | Inverse agonist | experimental | Small molecule | CNR1 inverse agonist |
| cannabidiol (Epidiolex) | Negative allosteric modulator | approved | Small molecule | CNR1 negative allosteric modulator |
| nimacimab | Negative allosteric modulator | experimental | mAb | Cannabinoid CB1 receptor negative allosteric modulator |
| omar | Radiopharmaceutical | experimental | Small molecule | CNR1 radiopharmaceutical |