← Mechanisms of action
RORC
SINGLE PROTEINHomo sapiens
Preferred name: Nuclear receptor ROR-gamma ChEMBL ↗
Linked proteins
Drugs acting on this target (23)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| lyc-55716 | Agonist | experimental | Small molecule | RORC agonist |
| rta 1701 | Allosteric antagonist | experimental | Small molecule | RORC allosteric antagonist |
| bi 730357 | Antagonist | experimental | Small molecule | RORC antagonist |
| jte-151 | Antagonist | experimental | Small molecule | RORC antagonist |
| jte-451 | Antagonist | experimental | Small molecule | RORC antagonist |
| abbv-553 | Inhibitor | experimental | Small molecule | RORC inhibitor |
| agn-242428 | Inhibitor | experimental | Small molecule | RORC inhibitor |
| arn-6039 | Inhibitor | experimental | Small molecule | RORC inhibitor |
| bos172767 | Inhibitor | experimental | Small molecule | RORC inhibitor |
| esr-114 | Inhibitor | experimental | Small molecule | RORC inhibitor |
| vtp-43742 | Inhibitor | experimental | Small molecule | RORC inhibitor |
| aur101 | Inverse agonist | experimental | Small molecule | RORC inverse agonist |
| azd0284 | Inverse agonist | experimental | Small molecule | RORC inverse agonist |
| azd4248 | Inverse agonist | experimental | Small molecule | RORC inverse agonist |
| bms-986251 | Inverse agonist | experimental | Small molecule | RORC inverse agonist |
| Cedirogant | Inverse agonist | experimental | Small molecule | RORC inverse agonist |
| gsk2981278 | Inverse agonist | experimental | Small molecule | RORC inverse agonist |
| imu-935 | Inverse agonist | experimental | Small molecule | RORC inverse agonist |
| jnj-61803534 | Inverse agonist | experimental | Small molecule | RORC inverse agonist |
| pf-06763809 | Inverse agonist | experimental | Small molecule | RORC inverse agonist |
| tak-828 | Inverse agonist | experimental | Small molecule | RORC inverse agonist |
| xj101 | Inverse agonist | experimental | Small molecule | RORC inverse agonist |
| xt-0528 | Inverse agonist | experimental | Small molecule | RORC inverse agonist |