← Mechanisms of action

RXFP1

SINGLE PROTEINHomo sapiens
Preferred name: Relaxin receptor 1 ChEMBL ↗

Linked proteins

Drugs acting on this target (9)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
f373280ActivatorexperimentalSmall moleculeRXFP1 activator
serelaxinActivatorexperimentalRecombinant proteinRXFP1 activator
azd5462AgonistexperimentalSmall moleculeRXFP1 agonist
frf-001AgonistexperimentalSmall moleculeRXFP1 agonist
ly3540378AgonistexperimentalSmall moleculeRXFP1 agonist
r2r01AgonistexperimentalSmall moleculeRXFP1 agonist
tx000045AgonistexperimentalSmall moleculeRXFP1 agonist
azd3427InhibitorexperimentalSmall moleculeRXFP1 inhibitor
mrna-0184SupplementationexperimentalNucleic acidRXFP1 supplementation