← Mechanisms of action
MAPT
SINGLE PROTEINHomo sapiens
Preferred name: Microtubule-associated protein tau ChEMBL ↗
Linked proteins
Drugs acting on this target (49)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| apnmab005 | Antagonist | experimental | mAb | Tau |
| nio752 | Antagonist | experimental | Small molecule | tau |
| aln-5288 | Antisense inhibitor | experimental | Nucleic acid | MAPT antisense inhibitor |
| aro-mapt-sc | Antisense inhibitor | experimental | Nucleic acid | MAPT antisense inhibitor |
| biib080 | Antisense inhibitor | experimental | Nucleic acid | tau |
| ionis maptrx | Antisense inhibitor | experimental | Nucleic acid | MAPT antisense inhibitor |
| [f-18]flornaptitril | Binding agent | experimental | Small molecule | MAPT binding agent |
| 18f-jss20-183a | Binding agent | experimental | Small molecule | MAPT binding agent |
| flortaucipir (Tauvid) | Binding agent | approved | Small molecule | MAPT binding agent |
| mni-815 | Binding agent | experimental | Small molecule | MAPT binding agent |
| ro-948 | Binding agent | experimental | Small molecule | Tau |
| ro6924963 | Binding agent | experimental | Small molecule | MAPT binding agent |
| ro6931643 | Binding agent | experimental | Small molecule | MAPT binding agent |
| t807 | Binding agent | experimental | Small molecule | MAPT binding agent |
| aadvac1 | Immunity, active | experimental | Vaccine | MAPT immunity, active |
| aci-35.030 | Immunity, active | experimental | Vaccine | MAPT immunity, active |
| av-1980r | Immunity, active | experimental | Vaccine | MAPT immunity, active |
| duvax | Immunity, active | experimental | Vaccine | MAPT immunity, active |
| jaci-35.054 | Immunity, active | experimental | Biological | MAPT immunity, active |
| protollin | Immunity, active | experimental | Vaccine | MAPT immunity, active |
| abbv-8e12 | Inhibitor | experimental | mAb | MAPT inhibitor |
| abbv-964i | Inhibitor | experimental | Small molecule | MAPT inhibitor |
| abbv-965i | Inhibitor | experimental | Small molecule | MAPT inhibitor |
| adel-y01 | Inhibitor | experimental | Small molecule | MAPT inhibitor |
| bey2153 | Inhibitor | experimental | Small molecule | MAPT inhibitor |
| biib061 | Inhibitor | experimental | Small molecule | MAPT inhibitor |
| biib076 | Inhibitor | experimental | mAb | MAPT inhibitor |
| bms-241027 | Inhibitor | experimental | Small molecule | MAPT inhibitor |
| bms-986168 | Inhibitor | experimental | mAb | MAPT inhibitor |
| da-7503 | Inhibitor | experimental | Small molecule | MAPT inhibitor |
| davunetide | Inhibitor | experimental | Peptide | MAPT inhibitor |
| dnl628 | Inhibitor | experimental | Small molecule | MAPT inhibitor |
| e2814 | Inhibitor | experimental | mAb | MAPT inhibitor |
| Hydromethylthionine | Inhibitor | experimental | Small molecule | MAPT inhibitor |
| jnj-63733657 | Inhibitor | experimental | mAb | MAPT inhibitor |
| jnj-64326067 | Inhibitor | experimental | Small molecule | MAPT inhibitor |
| lu af87908 | Inhibitor | experimental | mAb | MAPT inhibitor |
| ly3303560 | Inhibitor | experimental | mAb | MAPT inhibitor |
| mk-2214 | Inhibitor | experimental | mAb | MAPT inhibitor |
| olx-07010 | Inhibitor | experimental | Small molecule | MAPT inhibitor |
| pnt001 | Inhibitor | experimental | mAb | MAPT inhibitor |
| rem0046127 | Inhibitor | experimental | Small molecule | MAPT inhibitor |
| ro6926496 | Inhibitor | experimental | mAb | MAPT inhibitor |
| semorinemab | Inhibitor | experimental | mAb | Microtubule-associated protein tau inhibitor |
| trx0037 | Inhibitor | experimental | Small molecule | MAPT inhibitor |
| ucb0107 | Inhibitor | experimental | mAb | Microtubule-associated protein tau inhibitor |
| Florzolotau | Radiopharmaceutical | experimental | Small molecule | MAPT radiopharmaceutical |
| ro6958948 | Radiopharmaceutical | experimental | Small molecule | MAPT radiopharmaceutical |
| xtr006 | Radiopharmaceutical | experimental | Small molecule | MAPT radiopharmaceutical |