← Mechanisms of action

FKBP1A

SINGLE PROTEINHomo sapiens
Preferred name: FK506-binding protein 1A ChEMBL ↗

Linked proteins

Drugs acting on this target (8)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
everolimus (zortress)InhibitorapprovedSmall moleculeFKBP1A inhibitor
olocrolimusInhibitorexperimentalSmall moleculeFKBP1A inhibitor
pimecrolimus (elidel)InhibitorapprovedSmall moleculeFKBP1A inhibitor
sirolimus (rapamune)InhibitorapprovedSmall moleculeFKBP1A inhibitor
tacrolimus (prograf)InhibitorapprovedSmall moleculeFKBP1A inhibitor
temsirolimus (torisel)InhibitorapprovedSmall moleculeFKBP1A inhibitor
zotarolimusInhibitorexperimentalSmall moleculeFK506-binding protein 1A inhibitor
s48168StabiliserexperimentalSmall moleculeFKBP1A stabiliser