← Mechanisms of action
AHR
SINGLE PROTEINHomo sapiens
Preferred name: Aryl hydrocarbon receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (7)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| afp464 | Activator | experimental | Small molecule | AHR activator |
| tapinarof (Vtama) | Agonist | approved | Small molecule | AHR agonist |
| yuq-a1007 | Agonist | experimental | Small molecule | AHR agonist |
| bay2416964 | Antagonist | experimental | Small molecule | AHR antagonist |
| ik-175 | Antagonist | experimental | Small molecule | AHR |
| da-4505 | Inhibitor | experimental | Small molecule | AHR inhibitor |
| kyn-175 | Inhibitor | experimental | Small molecule | AHR inhibitor |