← Mechanisms of action

DHFR

SINGLE PROTEINHomo sapiens
Preferred name: Dihydrofolate reductase ChEMBL ↗

Linked proteins

Drugs acting on this target (6)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
aminopterinInhibitorexperimentalSmall moleculeDHFR inhibitor
methotrexateInhibitorexperimentalSmall moleculeDHFR inhibitor
naltrexone (revia)InhibitorapprovedSmall moleculeDHFR inhibitor
pemetrexed (alimta)InhibitorapprovedSmall moleculeDHFR inhibitor
piritreximInhibitorexperimentalSmall moleculeDihydrofolate reductase inhibitor
pralatrexate (folotyn)InhibitorapprovedSmall moleculeDHFR inhibitor