← Mechanisms of action
GHR
SINGLE PROTEINHomo sapiens
Preferred name: Growth hormone receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (14)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| eftansomatropin alfa | Agonist | experimental | Recombinant protein | GHR agonist |
| growth hormone (Protropin) | Agonist | approved | Biological | GHR agonist |
| ipamorelin | Agonist | experimental | Small molecule | GHR agonist |
| lat8881 | Agonist | experimental | Small molecule | GHR agonist |
| lonapegsomatropin (Skytrofa) | Agonist | approved | Recombinant protein | GHR agonist |
| mk-gh-04 | Agonist | experimental | Recombinant protein | GHR agonist |
| pegvisomant (somavert) | Agonist | approved | Recombinant protein | GHR agonist |
| somapacitan (Sogroya) | Agonist | approved | Small molecule | GHR agonist |
| somatrogon (Ngenla) | Agonist | approved | Recombinant protein | GHR agonist |
| somatropin (protropin) | Agonist | approved | Recombinant protein | GHR agonist |
| alxn2420 | Antagonist | experimental | Small molecule | GHR antagonist |
| mar002 | Antagonist | experimental | Small molecule | GHR antagonist |
| pegvisomant (somavert) | Antagonist | approved | Recombinant protein | GHR antagonist |
| ionis ghr-lrx | Inhibitor | experimental | Nucleic acid | GHR inhibitor |