← Mechanisms of action

ACVR2A

SINGLE PROTEINHomo sapiens
Preferred name: Activin receptor type-2A ChEMBL ↗

Linked proteins

Drugs acting on this target (8)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
imc-003ActivatorexperimentalRecombinant proteinACVR2A activator
bone morphogenetic protein-2AgonistexperimentalRecombinant proteinActivin receptor type-2A agonist
azd1043InhibitorexperimentalSmall moleculeACVR2A inhibitor
hs135InhibitorexperimentalRecombinant proteinACVR2A inhibitor
ker-012InhibitorexperimentalRecombinant proteinACVR2A inhibitor
lae102InhibitorexperimentalSmall moleculeACVR2A inhibitor
lae103InhibitorexperimentalmAbACVR2A inhibitor
sotatercept (WINREVAIR)InhibitorapprovedRecombinant proteinACVR2A inhibitor