← Mechanisms of action
SMO
SINGLE PROTEINHomo sapiens
Preferred name: Smoothened homolog ChEMBL ↗
Linked proteins
Drugs acting on this target (9)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| bms-833923 | Antagonist | experimental | Small molecule | SMO antagonist |
| glasdegib (Daurismo) | Antagonist | approved | Small molecule | SMO antagonist |
| leq-506 | Antagonist | experimental | Small molecule | SMO antagonist |
| tak-441 | Antagonist | experimental | Small molecule | SMO antagonist |
| taladegib | Antagonist | experimental | Small molecule | SMO antagonist |
| zsp1602 | Antagonist | experimental | Small molecule | SMO antagonist |
| saridegib | Inhibitor | experimental | Small molecule | SMO inhibitor |
| sonidegib (odomzo) | Inhibitor | approved | Small molecule | SMO inhibitor |
| vismodegib (erivedge) | Inhibitor | approved | Small molecule | SMO inhibitor |