← Mechanisms of action
HCAR2
SINGLE PROTEINHomo sapiens
Preferred name: Hydroxycarboxylic acid receptor 2 ChEMBL ↗
Linked proteins
Drugs acting on this target (7)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| acipimox | Agonist | experimental | Small molecule | HCAR2 agonist |
| gsk256073 | Agonist | experimental | Small molecule | HCAR2 agonist |
| mk1903 | Agonist | experimental | Small molecule | HCAR2 agonist |
| sch-900271 | Agonist | experimental | Small molecule | Hydroxycarboxylic acid receptor 2 agonist |
| lobeline | Antagonist | experimental | Small molecule | HCAR2 antagonist |
| sch 900271 | Inhibitor | experimental | Small molecule | HCAR2 inhibitor |
| mk0354 | Partial agonist | experimental | Small molecule | HCAR2 partial agonist |