← Mechanisms of action
GIPR
SINGLE PROTEINHomo sapiens
Preferred name: Gastric inhibitory polypeptide receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (28)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| bgm0504 | Agonist | experimental | Peptide | GIPR agonist |
| dulaglutide (trulicity) | Agonist | approved | Peptide | Gastric inhibitory polypeptide receptor agonist |
| gip | Agonist | experimental | Peptide | GIPR agonist |
| gip (3-30) | Agonist | experimental | Peptide | GIPR agonist |
| glp-1 (7-36) amide | Agonist | experimental | Peptide | GIPR agonist |
| gma106 | Agonist | experimental | mAb | GIPR agonist |
| hec-007 | Agonist | experimental | Peptide | GIPR agonist |
| hm15275 | Agonist | experimental | Peptide | GIPR agonist |
| hrs-4729 | Agonist | experimental | Peptide | GIPR agonist |
| hrs-9531 | Agonist | experimental | Peptide | GIPR agonist |
| hrs9531 | Agonist | experimental | Recombinant protein | GIPR agonist |
| kai-9531 | Agonist | experimental | Small molecule | GIPR agonist |
| ly3532226 | Agonist | experimental | Small molecule | GIPR agonist |
| ly3537021 | Agonist | experimental | Small molecule | GIPR agonist |
| mbx 4291 | Agonist | experimental | Peptide | GIPR agonist |
| mwn109 | Agonist | experimental | Peptide | GIPR agonist |
| na-931 | Agonist | experimental | Small molecule | GIPR agonist |
| nnc0480-0389 | Agonist | experimental | Small molecule | GIPR agonist |
| nnc9204-1706 a | Agonist | experimental | Peptide | GIPR agonist |
| pf-07940369 | Agonist | experimental | Small molecule | GIPR agonist |
| ro6807952 | Agonist | experimental | Small molecule | GIPR agonist |
| ro6811135 | Agonist | experimental | Peptide | GIPR agonist |
| thdbh120 | Agonist | experimental | Peptide | GIPR agonist |
| tirzepatide (Mounjaro) | Agonist | approved | Peptide | GIPR agonist |
| ubt251 | Agonist | experimental | Peptide | GIPR agonist |
| vk2735 | Agonist | experimental | Peptide | GIPR agonist |
| alv-100 | Antagonist | experimental | Peptide | GIPR antagonist |
| maridebart cafraglutide | Antagonist | experimental | Peptide | GIPR antagonist |