← Mechanisms of action

GIPR

SINGLE PROTEINHomo sapiens
Preferred name: Gastric inhibitory polypeptide receptor ChEMBL ↗

Linked proteins

Drugs acting on this target (28)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
bgm0504AgonistexperimentalPeptideGIPR agonist
dulaglutide (trulicity)AgonistapprovedPeptideGastric inhibitory polypeptide receptor agonist
gipAgonistexperimentalPeptideGIPR agonist
gip (3-30)AgonistexperimentalPeptideGIPR agonist
glp-1 (7-36) amideAgonistexperimentalPeptideGIPR agonist
gma106AgonistexperimentalmAbGIPR agonist
hec-007AgonistexperimentalPeptideGIPR agonist
hm15275AgonistexperimentalPeptideGIPR agonist
hrs-4729AgonistexperimentalPeptideGIPR agonist
hrs-9531AgonistexperimentalPeptideGIPR agonist
hrs9531AgonistexperimentalRecombinant proteinGIPR agonist
kai-9531AgonistexperimentalSmall moleculeGIPR agonist
ly3532226AgonistexperimentalSmall moleculeGIPR agonist
ly3537021AgonistexperimentalSmall moleculeGIPR agonist
mbx 4291AgonistexperimentalPeptideGIPR agonist
mwn109AgonistexperimentalPeptideGIPR agonist
na-931AgonistexperimentalSmall moleculeGIPR agonist
nnc0480-0389AgonistexperimentalSmall moleculeGIPR agonist
nnc9204-1706 aAgonistexperimentalPeptideGIPR agonist
pf-07940369AgonistexperimentalSmall moleculeGIPR agonist
ro6807952AgonistexperimentalSmall moleculeGIPR agonist
ro6811135AgonistexperimentalPeptideGIPR agonist
thdbh120AgonistexperimentalPeptideGIPR agonist
tirzepatide (Mounjaro)AgonistapprovedPeptideGIPR agonist
ubt251AgonistexperimentalPeptideGIPR agonist
vk2735AgonistexperimentalPeptideGIPR agonist
alv-100AntagonistexperimentalPeptideGIPR antagonist
maridebart cafraglutideAntagonistexperimentalPeptideGIPR antagonist