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Ferriprotoporphyrin IX

SMALL MOLECULEPlasmodium falciparum

Drugs acting on this target (12)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
hexyl 5-aminolevulinate (Cysview)ActivatorapprovedSmall moleculeFerriprotoporphyrin IX activator
aminolevulinic acid (levulan)AgonistapprovedSmall moleculeFerriprotoporphyrin IX agonist
dihydroartemisininBinding agentexperimentalSmall moleculeFerriprotoporphyrin IX binding agent
amodiaquine (camoquin)InhibitorapprovedSmall moleculeFerriprotoporphyrin IX inhibitor
artemetherInhibitorapprovedSmall moleculeFerriprotoporphyrin IX inhibitor
chloroquineInhibitorapprovedSmall moleculeFerriprotoporphyrin IX inhibitor
halofantrine (halfan)InhibitorapprovedSmall moleculeFerriprotoporphyrin IX inhibitor
hydroxychloroquine (plaquenil)InhibitorapprovedSmall moleculeFerriprotoporphyrin IX inhibitor
lumefantrine (Coartem)InhibitorapprovedSmall moleculeFerriprotoporphyrin IX inhibitor
mefloquine (lariam)InhibitorapprovedSmall moleculeFerriprotoporphyrin IX inhibitor
piperaquineInhibitorexperimentalSmall moleculeFerriprotoporphyrin IX inhibitor
quinine (qualaquin)InhibitorapprovedSmall moleculeFerriprotoporphyrin IX inhibitor