← Mechanisms of action
NR3C2
SINGLE PROTEINHomo sapiens
Preferred name: Mineralocorticoid receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (18)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| desoxycorticosterone pivalate | Agonist | approved | Small molecule | NR3C2 agonist |
| fludrocortisone (florinef) | Agonist | approved | Small molecule | NR3C2 agonist |
| Methoxypregnenolone | Agonist | experimental | Small molecule | NR3C2 agonist |
| canrenone (Contaren) | Antagonist | experimental | Small molecule | NR3C2 antagonist |
| drospirenone (Yasmin) | Antagonist | approved | Small molecule | NR3C2 antagonist |
| eplerenone (inspra) | Antagonist | approved | Small molecule | NR3C2 antagonist |
| esaxerenone | Antagonist | experimental | Small molecule | NR3C2 antagonist |
| felodipine (plendil) | Antagonist | approved | Small molecule | NR3C2 antagonist |
| finerenone (KERENDIA) | Antagonist | approved | Small molecule | NR3C2 antagonist |
| hrs-2183 | Antagonist | experimental | Small molecule | NR3C2 antagonist |
| ly2623091 | Antagonist | experimental | Small molecule | NR3C2 antagonist |
| mt-3995 | Antagonist | experimental | Small molecule | NR3C2 antagonist |
| nimodipine (nimotop) | Antagonist | approved | Small molecule | NR3C2 antagonist |
| Ocedurenone | Antagonist | experimental | Small molecule | NR3C2 antagonist |
| pf-03882845 | Antagonist | experimental | Small molecule | NR3C2 antagonist |
| spironolactone (aldactone) | Antagonist | approved | Small molecule | NR3C2 antagonist |
| vamorolone (Agamree) | Antagonist | approved | Small molecule | NR3C2 antagonist |
| Balcinrenone | Modulator | experimental | Small molecule | NR3C2 modulator |