← Mechanisms of action
FGFR1
SINGLE PROTEINHomo sapiens
Preferred name: Fibroblast growth factor receptor 1 ChEMBL ↗
Linked proteins
Drugs acting on this target (55)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| nx-13 | Activator | experimental | Small molecule | FGFR1 activator |
| fgf-21 | Agonist | experimental | Recombinant protein | FGFR1 agonist |
| hec88473 | Agonist | experimental | Recombinant protein | FGFR1 agonist |
| jmt202 | Agonist | experimental | Small molecule | FGFR1 agonist |
| ly3025876 | Agonist | experimental | Small molecule | FGFR1 agonist |
| ly3084077 | Agonist | experimental | Small molecule | FGFR1 agonist |
| nnc0194-0499 | Agonist | experimental | Small molecule | FGFR1 agonist |
| sun13837 | Agonist | experimental | Small molecule | FGFR1 agonist |
| kin-3248 | Antagonist | experimental | Small molecule | FGFR1 antagonist |
| tt-00434 | Antagonist | experimental | Small molecule | FGFR1 antagonist |
| 3d185 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| absk091 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| absk121 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| al8326 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| anrotenib | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| asp5878 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| aur109 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| azd4547 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| bfkb8488a | Inhibitor | experimental | mAb | FGFR1 inhibitor |
| bt01001 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| ch5183284 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| chir-258 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| cpl304110 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| debio-1347 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| derazantinib | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| e7090 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| eoc317 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| esk981 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| et0111 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| Gunagratinib | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| imlifidase | Inhibitor | experimental | Recombinant protein | Fibroblast growth factor receptor 1 inhibitor |
| inca00186 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| lucitanib | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| ly4298445 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| max-40279 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| mk-3655 | Inhibitor | experimental | mAb | FGFR1 inhibitor |
| nindetanib | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| odm 203 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| odm-203 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| om-rca-01 | Inhibitor | experimental | mAb | FGFR1 inhibitor |
| pazopanib (votrient) | Inhibitor | approved | Small molecule | FGFR1 inhibitor |
| pemigatinib (Pemazyre) | Inhibitor | approved | Small molecule | Fibroblast growth factor receptor 1 inhibitor |
| Pimicotinib | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| prn1371 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| regorafenib (stivarga) | Inhibitor | approved | Small molecule | FGFR1 inhibitor |
| rg002 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| rg1530 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| simmitinib | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| sulfatinib | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| surufatinib | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| tcmdc-140940 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| tg-100801 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| Tinengotinib | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| tyra-200 | Inhibitor | experimental | Small molecule | FGFR1 inhibitor |
| aav9 bbp-812 | Supplementation | experimental | Gene therapy | FGFR1 supplementation |