← Mechanisms of action
FGFR2
SINGLE PROTEINHomo sapiens
Preferred name: Fibroblast growth factor receptor 2 ChEMBL ↗
Linked proteins
Drugs acting on this target (45)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| ly3025876 | Agonist | experimental | Small molecule | FGFR2 agonist |
| ly3084077 | Agonist | experimental | Small molecule | FGFR2 agonist |
| palifermin (Kepivance) | Agonist | approved | Recombinant protein | FGFR2 agonist |
| trafermin | Agonist | experimental | Recombinant protein | FGFR2 agonist |
| absk061 | Antagonist | experimental | Small molecule | FGFR2 antagonist |
| bemarituzumab | Antagonist | experimental | mAb | Fibroblast growth factor receptor 2 antagonist |
| erdafitinib (Balversa) | Antagonist | approved | Small molecule | FGFR2 antagonist |
| futibatinib (Lytgobi) | Antagonist | approved | Small molecule | FGFR2 antagonist |
| pemigatinib (Pemazyre) | Antagonist | approved | Small molecule | FGFR2 antagonist |
| tt-00434 | Antagonist | experimental | Small molecule | FGFR2 antagonist |
| 3d185 | Inhibitor | experimental | Small molecule | FGFR2 inhibitor |
| 3h-10000 | Inhibitor | experimental | mAb | FGFR2 inhibitor |
| 3hp-2827 | Inhibitor | experimental | Small molecule | FGFR2 inhibitor |
| absk091 | Inhibitor | experimental | Small molecule | FGFR2 inhibitor |
| absk121 | Inhibitor | experimental | Small molecule | FGFR2 inhibitor |
| alofanib | Inhibitor | experimental | Small molecule | FGFR2 inhibitor |
| anrotenib | Inhibitor | experimental | Small molecule | FGFR2 inhibitor |
| asp5878 | Inhibitor | experimental | Small molecule | FGFR2 inhibitor |
| azd4547 | Inhibitor | experimental | Small molecule | FGFR2 inhibitor |
| bay1179470 | Inhibitor | experimental | mAb | FGFR2 inhibitor |
| bay1187982 | Inhibitor | experimental | mAb | FGFR2 inhibitor |
| bemarituzumab | Inhibitor | experimental | mAb | FGFR2 inhibitor |
| bg-c137 | Inhibitor | experimental | mAb | FGFR2 inhibitor |
| cgt4859 | Inhibitor | experimental | Small molecule | FGFR2 inhibitor |
| cpl304110 | Inhibitor | experimental | Small molecule | FGFR2 inhibitor |
| debio-1347 | Inhibitor | experimental | Small molecule | FGFR2 inhibitor |
| derazantinib | Inhibitor | experimental | Small molecule | FGFR2 inhibitor |
| ds-1123 | Inhibitor | experimental | mAb | FGFR2 inhibitor |
| et0111 | Inhibitor | experimental | Small molecule | FGFR2 inhibitor |
| Gunagratinib | Inhibitor | experimental | Small molecule | FGFR2 inhibitor |
| hdm2020 | Inhibitor | experimental | mAb | FGFR2 inhibitor |
| imlifidase | Inhibitor | experimental | Recombinant protein | Fibroblast growth factor receptor 2 inhibitor |
| inca00186 | Inhibitor | experimental | Small molecule | FGFR2 inhibitor |
| knt-0916 | Inhibitor | experimental | Small molecule | FGFR2 inhibitor |
| lucitanib | Inhibitor | experimental | Small molecule | FGFR2 inhibitor |
| ly4298445 | Inhibitor | experimental | Small molecule | FGFR2 inhibitor |
| pemigatinib (Pemazyre) | Inhibitor | approved | Small molecule | Fibroblast growth factor receptor 2 inhibitor |
| regorafenib (stivarga) | Inhibitor | approved | Small molecule | FGFR2 inhibitor |
| rg002 | Inhibitor | experimental | Small molecule | FGFR2 inhibitor |
| rg1530 | Inhibitor | experimental | Small molecule | FGFR2 inhibitor |
| rly-4008 | Inhibitor | experimental | Small molecule | FGFR2 inhibitor |
| sim0686 | Inhibitor | experimental | mAb | FGFR2 inhibitor |
| tg-100801 | Inhibitor | experimental | Small molecule | FGFR2 inhibitor |
| tqb2210 | Inhibitor | experimental | Small molecule | FGFR2 inhibitor |
| tyra-200 | Inhibitor | experimental | Small molecule | FGFR2 inhibitor |