← Mechanisms of action
DNMT1
SINGLE PROTEINHomo sapiens
Preferred name: DNA (cytosine-5)-methyltransferase 1 ChEMBL ↗
Linked proteins
Drugs acting on this target (9)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| mg98 | Antisense inhibitor | experimental | Nucleic acid | DNMT1 antisense inhibitor |
| ntx-301 | Antisense inhibitor | experimental | Nucleic acid | DNMT1 antisense inhibitor |
| 5-Aza-4'-thio-2'-deoxycytidine | Inhibitor | experimental | Small molecule | DNMT1 inhibitor |
| azacitidine (vidaza) | Inhibitor | approved | Small molecule | DNMT1 inhibitor |
| decitabine (dacogen) | Inhibitor | approved | Small molecule | DNMT1 inhibitor |
| ef-009 | Inhibitor | experimental | Small molecule | DNMT1 inhibitor |
| gsk4172239d | Inhibitor | experimental | Small molecule | DNMT1 inhibitor |
| guadecitabine | Inhibitor | experimental | Small molecule | DNMT1 inhibitor |
| larsucosterol | Inhibitor | experimental | Small molecule | DNMT1 inhibitor |