← Mechanisms of action
MPL
SINGLE PROTEINHomo sapiens
Preferred name: Thrombopoietin receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (9)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| ono-7746 | Activator | experimental | Small molecule | MPL activator |
| avatrombopag | Agonist | approved | Small molecule | MPL agonist |
| eltrombopag (promacta) | Agonist | approved | Small molecule | MPL agonist |
| hetrombopag olamine | Agonist | experimental | Small molecule | MPL agonist |
| lgd-4665 | Agonist | experimental | Small molecule | MPL agonist |
| Lusutrombopag (Mulpleta) | Agonist | approved | Small molecule | MPL agonist |
| pn20 | Agonist | experimental | Small molecule | MPL agonist |
| romiplostim (nplate) | Agonist | approved | Small molecule | MPL agonist |
| inca033989 | Inhibitor | experimental | mAb | MPL inhibitor |