← Mechanisms of action

PTGER4

SINGLE PROTEINHomo sapiens
Preferred name: Prostanoid EP4 receptor ChEMBL ↗

Linked proteins

Drugs acting on this target (16)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
rivenprostAgonistexperimentalSmall moleculePTGER4 agonist
asp7657AntagonistexperimentalSmall moleculePTGER4 antagonist
bgc20-1531AntagonistexperimentalSmall moleculePTGER4 antagonist
bms-986310AntagonistexperimentalSmall moleculePTGER4 antagonist
dcby02AntagonistexperimentalmAbPTGER4 antagonist
dt-9081AntagonistexperimentalSmall moleculePTGER4 antagonist
e7046AntagonistexperimentalSmall moleculePTGER4 antagonist
grapiprantAntagonistexperimentalSmall moleculeProstanoid EP4 receptor antagonist
ono-4578AntagonistexperimentalSmall moleculePTGER4 antagonist
an0025InhibitorexperimentalSmall moleculePTGER4 inhibitor
cr6086InhibitorexperimentalSmall moleculePTGER4 inhibitor
grapiprantInhibitorexperimentalSmall moleculePTGER4 inhibitor
inv-1120InhibitorexperimentalSmall moleculePTGER4 inhibitor
ly3127760InhibitorexperimentalSmall moleculePTGER4 inhibitor
mbf-362InhibitorexperimentalSmall moleculePTGER4 inhibitor
tpst-1495InhibitorexperimentalSmall moleculePTGER4 inhibitor