← Mechanisms of action
NPR1
SINGLE PROTEINHomo sapiens
Preferred name: Atrial natriuretic peptide receptor A ChEMBL ↗
Linked proteins
Drugs acting on this target (25)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| avenciguat | Activator | experimental | Small molecule | NPR1 activator |
| bay1211163 | Activator | experimental | Small molecule | NPR1 activator |
| iw-6463 | Activator | experimental | Small molecule | NPR1 activator |
| manp | Activator | experimental | Peptide | NPR1 activator |
| mgv354 | Activator | experimental | Small molecule | NPR1 activator |
| mk-5475 | Activator | experimental | Small molecule | NPR1 activator |
| mosliciguat | Activator | experimental | Small molecule | NPR1 activator |
| nitric acid | Activator | experimental | Small molecule | NPR1 activator |
| plecanatide (trulance) | Activator | approved | Peptide | NPR1 activator |
| praliciguat | Activator | experimental | Small molecule | NPR1 activator |
| runcaciguat | Activator | experimental | Small molecule | NPR1 activator |
| urodilatin | Activator | experimental | Small molecule | NPR1 activator |
| linaclotide (linzess) | Agonist | approved | Peptide | NPR1 agonist |
| Nelociguat | Agonist | experimental | Small molecule | NPR1 agonist |
| nesiritide (natrecor) | Agonist | approved | Peptide | NPR1 agonist |
| pl-3994 | Agonist | experimental | Small molecule | Atrial natriuretic peptide receptor A agonist |
| pl3994 | Agonist | experimental | Small molecule | NPR1 agonist |
| REGN9035 | Antagonist | experimental | mAb | NPR1 |
| bay1101042 | Inhibitor | experimental | Small molecule | NPR1 inhibitor |
| bay3283142 | Inhibitor | experimental | Small molecule | NPR1 inhibitor |
| regn5381 | Inhibitor | experimental | mAb | NPR1 inhibitor |
| regn7544 | Inhibitor | experimental | mAb | NPR1 inhibitor |
| regn7544 | Inhibitor | experimental | mAb | NPR1 inhibitor |
| xxb750 | Inhibitor | experimental | Small molecule | NPR1 inhibitor |
| zagociguat | Inhibitor | experimental | Small molecule | NPR1 inhibitor |