← Mechanisms of action
CYP17A1
SINGLE PROTEINHomo sapiens
Preferred name: Cytochrome P450 17A1 ChEMBL ↗
Linked proteins
Drugs acting on this target (11)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| 17-deoxycortisol | Inhibitor | experimental | Small molecule | CYP17A1 inhibitor |
| abiraterone (zytiga) | Inhibitor | approved | Small molecule | CYP17A1 inhibitor |
| asn001 | Inhibitor | experimental | Small molecule | CYP17A1 inhibitor |
| cfg920 | Inhibitor | experimental | Small molecule | CYP17A1 inhibitor |
| ds-6000a | Inhibitor | experimental | mAb | CYP17A1 inhibitor |
| galeterone | Inhibitor | experimental | Small molecule | CYP17A1 inhibitor |
| ketoconazole (nizoral) | Inhibitor | approved | Small molecule | Cytochrome P450 17A1 inhibitor |
| lae001 | Inhibitor | experimental | Small molecule | CYP17A1 inhibitor |
| odm-204 | Inhibitor | experimental | Small molecule | CYP17A1 inhibitor |
| orteronel | Inhibitor | experimental | Small molecule | CYP17A1 inhibitor |
| seviteronel | Inhibitor | experimental | Small molecule | Cytochrome P450 17A1 inhibitor |