← Mechanisms of action

GRM2

SINGLE PROTEINHomo sapiens
Preferred name: Metabotropic glutamate receptor 2 ChEMBL ↗

Linked proteins

Drugs acting on this target (15)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
ly-404039AgonistexperimentalSmall moleculeGRM2 agonist
ly2300559AgonistexperimentalSmall moleculeGRM2 agonist
ly2969822AgonistexperimentalSmall moleculeGRM2 agonist
ly2979165AgonistexperimentalSmall moleculeGRM2 agonist
pomaglumetadAgonistexperimentalSmall moleculeGRM2 agonist
bci-1038AntagonistexperimentalSmall moleculeGRM2 antagonist
bci-1283AntagonistexperimentalSmall moleculeGRM2 antagonist
bci-838AntagonistexperimentalSmall moleculeGRM2 antagonist
gate-101AntagonistexperimentalSmall moleculeGRM2 antagonist
ts-161InhibitorexperimentalSmall moleculeGRM2 inhibitor
decoglurantModulatorexperimentalSmall moleculeGRM2 modulator
jnj-40411813ModulatorexperimentalSmall moleculeGRM2 modulator
jnj-55375515ModulatorexperimentalSmall moleculeGRM2 modulator
azd8529Positive allosteric modulatorexperimentalSmall moleculeGRM2 positive allosteric modulator
jnj-40411813Positive allosteric modulatorexperimentalSmall moleculeMetabotropic glutamate receptor 2 positive allosteric modulator