← Mechanisms of action
ADRB3
SINGLE PROTEINHomo sapiens
Preferred name: Beta-3 adrenergic receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (9)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| amibegron | Agonist | experimental | Small molecule | ADRB3 agonist |
| ly-377604 | Agonist | experimental | Small molecule | ADRB3 agonist |
| mirabegron (myrbetriq) | Agonist | approved | Small molecule | ADRB3 agonist |
| ritobegron | Agonist | experimental | Small molecule | ADRB3 agonist |
| solabegron | Agonist | experimental | Small molecule | ADRB3 agonist |
| tak-677 | Agonist | experimental | Small molecule | ADRB3 agonist |
| vibegron (Gemtesa) | Agonist | approved | Small molecule | ADRB3 agonist |
| apd418 | Inhibitor | experimental | Small molecule | ADRB3 inhibitor |
| cgp12177 | Partial agonist | experimental | Small molecule | ADRB3 partial agonist |