← Mechanisms of action
C5AR1
SINGLE PROTEINHomo sapiens
Preferred name: C5a anaphylatoxin chemotactic receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (15)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| act-1014-6470 | Antagonist | experimental | Small molecule | C5AR1 antagonist |
| avacopan (Tavneos) | Antagonist | approved | Small molecule | C5AR1 antagonist |
| mp-435 | Antagonist | experimental | Small molecule | C5AR1 antagonist |
| vis954 | Antagonist | experimental | Small molecule | C5AR1 antagonist |
| aon-d21 | Inhibitor | experimental | Nucleic acid | C5AR1 inhibitor |
| avdoralimab | Inhibitor | experimental | mAb | C5a anaphylatoxin chemotactic receptor inhibitor |
| bdb-001 | Inhibitor | experimental | mAb | C5AR1 inhibitor |
| can106 | Inhibitor | experimental | Small molecule | C5AR1 inhibitor |
| hib210 | Inhibitor | experimental | mAb | C5AR1 inhibitor |
| iph5401 | Inhibitor | experimental | mAb | C5AR1 inhibitor |
| kp104 | Inhibitor | experimental | mAb | C5AR1 inhibitor |
| nnc 0151-0000-0000 | Inhibitor | experimental | mAb | C5AR1 inhibitor |
| nnc0215-0384 | Inhibitor | experimental | mAb | C5AR1 inhibitor |
| stsa-1002 | Inhibitor | experimental | mAb | C5AR1 inhibitor |
| tj210001 | Inhibitor | experimental | mAb | C5AR1 inhibitor |