← Mechanisms of action
F10
SINGLE PROTEINHomo sapiens
Preferred name: Coagulation factor X ChEMBL ↗
Linked proteins
Drugs acting on this target (32)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| stsp-0601 | Activator | experimental | Animal product | F10 activator |
| human coagulation factor x (Coagadex) | Agonist | approved | Biological | F10 agonist |
| mim8 | Agonist | experimental | mAb | F10 agonist |
| rivaroxaban (xarelto) | Antagonist | approved | Small molecule | F10 antagonist |
| human coagulation factor x (Coagadex) | Exogenous protein | approved | Biological | Coagulation factor X exogenous protein |
| human factor ix complex (prothrombin complex concentrate) (Bebulin) | Exogenous protein | approved | Biological | Coagulation factor X exogenous protein |
| amblyomin-x | Inhibitor | experimental | Recombinant protein | F10 inhibitor |
| apixaban (eliquis) | Inhibitor | approved | Small molecule | F10 inhibitor |
| bay 3389934 | Inhibitor | experimental | Small molecule | F10 inhibitor |
| bay3389934 | Inhibitor | experimental | Small molecule | F10 inhibitor |
| bemiparin (Ivor) | Inhibitor | experimental | Small molecule | Coagulation factor X inhibitor |
| betrixaban (bevyxxa) | Inhibitor | approved | Small molecule | F10 inhibitor |
| bi 11634 | Inhibitor | experimental | Small molecule | F10 inhibitor |
| bibt 1011 bs | Inhibitor | experimental | Small molecule | F10 inhibitor |
| bibt 986 | Inhibitor | experimental | Small molecule | F10 inhibitor |
| ckd-344 | Inhibitor | experimental | Small molecule | F10 inhibitor |
| darexaban | Inhibitor | experimental | Small molecule | F10 inhibitor |
| Dimolegin | Inhibitor | experimental | Small molecule | F10 inhibitor |
| edoxaban (savaysa) | Inhibitor | approved | Small molecule | F10 inhibitor |
| gcc-4401 | Inhibitor | experimental | Small molecule | F10 inhibitor |
| gw813893 | Inhibitor | experimental | Peptide | F10 inhibitor |
| idraparinux | Inhibitor | experimental | Small molecule | F10 inhibitor |
| letaxaban | Inhibitor | experimental | Small molecule | F10 inhibitor |
| ly517717 | Inhibitor | experimental | Small molecule | F10 inhibitor |
| nxt007 | Inhibitor | experimental | mAb | F10 inhibitor |
| otamixaban | Inhibitor | experimental | Small molecule | F10 inhibitor |
| pd0348292 | Inhibitor | experimental | Small molecule | F10 inhibitor |
| ro-14 | Inhibitor | experimental | Small molecule | F10 inhibitor |
| syha136 | Inhibitor | experimental | Small molecule | F10 inhibitor |
| andexanet alfa (Andexxa) | Supplementation | experimental | Recombinant protein | F10 supplementation |
| pf-05230907 | Supplementation | experimental | Recombinant protein | F10 supplementation |
| vmx-c001 | Supplementation | experimental | Recombinant protein | F10 supplementation |