← Mechanisms of action

Q7ZJM1

SINGLE PROTEINHuman immunodeficiency virus 1
Preferred name: Human immunodeficiency virus type 1 integrase ChEMBL ↗

Linked proteins

Drugs acting on this target (15)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
cabotegravir (Vocabria)AntagonistapprovedSmall moleculeQ7ZJM1 antagonist
bi 224436InhibitorexperimentalSmall moleculeQ7ZJM1 inhibitor
bictegravir (Biktarvy)InhibitorapprovedSmall moleculeQ7ZJM1 inhibitor
bms-707035InhibitorexperimentalSmall moleculeQ7ZJM1 inhibitor
cabotegravir (Vocabria)InhibitorapprovedSmall moleculeHuman immunodeficiency virus type 1 integrase inhibitor
dolutegravir (tivicay)InhibitorapprovedSmall moleculeQ7ZJM1 inhibitor
elvitegravir (vitekta)InhibitorapprovedSmall moleculeQ7ZJM1 inhibitor
gsk-364735InhibitorexperimentalSmall moleculeHuman immunodeficiency virus type 1 integrase inhibitor
gsk364735InhibitorexperimentalSmall moleculeQ7ZJM1 inhibitor
gw810781InhibitorexperimentalSmall moleculeQ7ZJM1 inhibitor
mk-2048InhibitorexperimentalSmall moleculeQ7ZJM1 inhibitor
pf-04776548InhibitorexperimentalSmall moleculeQ7ZJM1 inhibitor
PirmitegravirInhibitorexperimentalSmall moleculeQ7ZJM1 inhibitor
raltegravir (isentress)InhibitorapprovedSmall moleculeQ7ZJM1 inhibitor
vh4524184InhibitorexperimentalSmall moleculeQ7ZJM1 inhibitor