← Mechanisms of action

P2RY12

SINGLE PROTEINHomo sapiens
Preferred name: Purinergic receptor P2Y12 ChEMBL ↗

Linked proteins

Drugs acting on this target (15)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
act-281959AntagonistexperimentalSmall moleculeP2RY12 antagonist
cangrelor (kengreal)AntagonistapprovedSmall moleculeP2RY12 antagonist
clopidogrel (plavix)AntagonistapprovedSmall moleculeP2RY12 antagonist
elinogrelAntagonistexperimentalSmall moleculeP2RY12 antagonist
prasugrel (effient)AntagonistapprovedSmall moleculeP2RY12 antagonist
regrelor disodiumAntagonistexperimentalSmall moleculeP2RY12 antagonist
selatogrelAntagonistexperimentalSmall moleculePurinergic receptor P2Y12 antagonist
ticagrelor (brilinta)AntagonistapprovedSmall moleculeP2RY12 antagonist
ticlopidine (ticlid)AntagonistapprovedSmall moleculeP2RY12 antagonist
thienoyridineImmunity, activeexperimentalSmall moleculeP2RY12 immunity, active
cangrelor (kengreal)InhibitorapprovedSmall moleculePurinergic receptor P2Y12 inhibitor
p2611222InhibitorexperimentalSmall moleculeP2RY12 inhibitor
selatogrelInhibitorexperimentalSmall moleculeP2RY12 inhibitor
tipidogrelInhibitorexperimentalSmall moleculeP2RY12 inhibitor
vicagrelInhibitorexperimentalSmall moleculeP2RY12 inhibitor