← Mechanisms of action
FGFR3
SINGLE PROTEINHomo sapiens
Preferred name: Fibroblast growth factor receptor 3 ChEMBL ↗
Linked proteins
Drugs acting on this target (35)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| ly3025876 | Agonist | experimental | Small molecule | FGFR3 agonist |
| ly3084077 | Agonist | experimental | Small molecule | FGFR3 agonist |
| ta-46 | Agonist | experimental | Recombinant protein | FGFR3 agonist |
| erdafitinib (Balversa) | Antagonist | approved | Small molecule | FGFR3 antagonist |
| loxo-435 | Antagonist | experimental | Small molecule | fgfr3 |
| pf-06755347 | Antagonist | experimental | mAb | FGFR3 antagonist |
| tt-00434 | Antagonist | experimental | Small molecule | FGFR3 antagonist |
| tyra-300 | Antagonist | experimental | Small molecule | fgfr3 |
| vosoritide (Voxzogo) | Antagonist | approved | Peptide | FGFR3 antagonist |
| 3d185 | Inhibitor | experimental | Small molecule | FGFR3 inhibitor |
| absk091 | Inhibitor | experimental | Small molecule | FGFR3 inhibitor |
| absk121 | Inhibitor | experimental | Small molecule | FGFR3 inhibitor |
| anrotenib | Inhibitor | experimental | Small molecule | FGFR3 inhibitor |
| azd4547 | Inhibitor | experimental | Small molecule | FGFR3 inhibitor |
| b-701 | Inhibitor | experimental | mAb | FGFR3 inhibitor |
| bhv-1530 | Inhibitor | experimental | mAb | FGFR3 inhibitor |
| cgt4859 | Inhibitor | experimental | Small molecule | FGFR3 inhibitor |
| cpl304110 | Inhibitor | experimental | Small molecule | FGFR3 inhibitor |
| debio-1347 | Inhibitor | experimental | Small molecule | FGFR3 inhibitor |
| derazantinib | Inhibitor | experimental | Small molecule | FGFR3 inhibitor |
| dovitinib | Inhibitor | experimental | Small molecule | FGFR3 inhibitor |
| enmd 2076 | Inhibitor | experimental | Small molecule | FGFR3 inhibitor |
| et0111 | Inhibitor | experimental | Small molecule | FGFR3 inhibitor |
| Gunagratinib | Inhibitor | experimental | Small molecule | FGFR3 inhibitor |
| imlifidase | Inhibitor | experimental | Recombinant protein | Fibroblast growth factor receptor 3 inhibitor |
| inca00186 | Inhibitor | experimental | Small molecule | FGFR3 inhibitor |
| ly3076226 | Inhibitor | experimental | mAb | FGFR3 inhibitor |
| masitinib | Inhibitor | experimental | Small molecule | FGFR3 inhibitor |
| pazopanib (votrient) | Inhibitor | approved | Small molecule | FGFR3 inhibitor |
| pemigatinib (Pemazyre) | Inhibitor | approved | Small molecule | Fibroblast growth factor receptor 3 inhibitor |
| rg-7444 | Inhibitor | experimental | mAb | FGFR3 inhibitor |
| sar442501 | Inhibitor | experimental | mAb | FGFR3 inhibitor |
| tyra-200 | Inhibitor | experimental | Small molecule | FGFR3 inhibitor |
| tyra-430 | Inhibitor | experimental | Small molecule | FGFR3 inhibitor |
| fpi-1966 | Radiodepletion | experimental | mAb | FGFR3 radiodepletion |