← Mechanisms of action
PTH1R
SINGLE PROTEINHomo sapiens
Preferred name: Parathyroid hormone receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (9)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| pco371 | Activator | experimental | Small molecule | PTH1R activator |
| abaloparatide (tymlos) | Agonist | approved | Peptide | PTH1R agonist |
| mbx 2109 | Agonist | experimental | Peptide | PTH1R agonist |
| palopegteriparatide (Yorvipath) | Agonist | approved | Peptide | Parathyroid hormone receptor agonist |
| parathyroid hormone (Natpara) | Agonist | approved | Recombinant protein | PTH1R agonist |
| teriparatide | Agonist | approved | Peptide | PTH1R agonist |
| zt-031 | Agonist | experimental | Small molecule | PTH1R agonist |
| azp-3601 | Antagonist | experimental | Peptide | Parathyroid hormone receptor |
| mt1013 | Antagonist | experimental | Peptide | PTH1R antagonist |