← Mechanisms of action

GSPT1

SINGLE PROTEINHomo sapiens
Preferred name: Eukaryotic peptide chain release factor GTP-binding subunit ERF3A ChEMBL ↗

Linked proteins

Drugs acting on this target (5)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
btx-1188DegraderexperimentalSmall moleculedegrader - GSPT1
cg009301DegraderexperimentalSmall moleculeGSPT1 degrader
ct-01DegraderexperimentalSmall moleculeGSPT1 degrader
mrt-2359DegraderexperimentalSmall moleculedegrader - GSPT1
fd-001InhibitorexperimentalSmall moleculeGSPT1 inhibitor