← Mechanisms of action
SCNN1A
SINGLE PROTEINHomo sapiens
Preferred name: Amiloride-sensitive sodium channel alpha-subunit ChEMBL ↗
Linked proteins
Drugs acting on this target (13)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| solnatide | Activator | experimental | Peptide | SCNN1A activator |
| ap301 | Agonist | experimental | Peptide | SCNN1A agonist |
| benzocaine (Orajel) | Antagonist | marketed | Small molecule | SCNN1A antagonist |
| gs-9411 | Antagonist | experimental | Small molecule | SCNN1A antagonist |
| qbw276 | Antisense inhibitor | experimental | Nucleic acid | SCNN1A antisense inhibitor |
| azd5634 | Inhibitor | experimental | Small molecule | SCNN1A inhibitor |
| bi 1265162 | Inhibitor | experimental | Small molecule | SCNN1A inhibitor |
| bi 443651 | Inhibitor | experimental | Small molecule | SCNN1A inhibitor |
| gs-5737 | Inhibitor | experimental | Small molecule | SCNN1A inhibitor |
| ionis-enacrx | Inhibitor | experimental | Nucleic acid | SCNN1A inhibitor |
| p-321 | Inhibitor | experimental | Small molecule | SCNN1A inhibitor |
| p-552 | Inhibitor | experimental | Small molecule | SCNN1A inhibitor |
| spx-101 | Inhibitor | experimental | Small molecule | SCNN1A inhibitor |