← Mechanisms of action
Cardiac myosin
PROTEIN COMPLEXHomo sapiens
Linked proteins
Drugs acting on this target (8)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| danicamtiv | Activator | experimental | Small molecule | Cardiac myosin activator |
| omecamtiv mecarbil | Activator | experimental | Small molecule | Cardiac myosin activator |
| mavacamten (Camzyos) | Antagonist | approved | Small molecule | Cardiac myosin antagonist |
| myk-224 | Antagonist | experimental | Small molecule | cardiac myosin |
| aficamten | Inhibitor | approved | Small molecule | Cardiac myosin inhibitor |
| ck-4021586 | Inhibitor | experimental | Small molecule | Cardiac myosin inhibitor |
| edg-5506 | Inhibitor | experimental | Small molecule | inhibitor - MYH7 |
| mavacamten (Camzyos) | Inhibitor | approved | Small molecule | Cardiac myosin inhibitor |