← Mechanisms of action

ABCB1

SINGLE PROTEINHomo sapiens
Preferred name: P-glycoprotein 1 ChEMBL ↗

Linked proteins

Drugs acting on this target (5)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
BIRICODARInhibitorexperimentalSmall moleculeP-glycoprotein 1 inhibitor
cyclosporine (sandimmune)InhibitorapprovedSmall moleculeP-glycoprotein 1 inhibitor
encequidarInhibitorexperimentalSmall moleculeABCB1 inhibitor
tariquidarInhibitorexperimentalSmall moleculeABCB1 inhibitor
zosuquidarInhibitorexperimentalSmall moleculeP-glycoprotein 1 inhibitor