← Mechanisms of action
AGTR1
SINGLE PROTEINHomo sapiens
Preferred name: Type-1 angiotensin II receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (21)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| c21 | Activator | experimental | Small molecule | AGTR1 activator |
| angiotensin ii | Agonist | approved | Peptide | AGTR1 agonist |
| mor107 | Agonist | experimental | Small molecule | AGTR1 agonist |
| trv027 | Agonist | experimental | Small molecule | AGTR1 agonist |
| azilsartan (edarbi) | Antagonist | approved | Small molecule | AGTR1 antagonist |
| candesartan (atacand) | Antagonist | approved | Small molecule | AGTR1 antagonist |
| ema400 | Antagonist | experimental | Small molecule | AGTR1 antagonist |
| eprosartan (teveten) | Antagonist | approved | Small molecule | AGTR1 antagonist |
| fimasartan (kanarb) | Antagonist | experimental | Small molecule | Type-1 angiotensin II receptor antagonist |
| irbesartan (avapro) | Antagonist | approved | Small molecule | AGTR1 antagonist |
| losartan (cozaar) | Antagonist | approved | Small molecule | AGTR1 antagonist |
| olmesartan (benicar) | Antagonist | approved | Small molecule | AGTR1 antagonist |
| qr12000 | Antagonist | experimental | Small molecule | AGTR1 antagonist |
| saralasin (sarenin) | Antagonist | approved | Small molecule | AGTR1 antagonist |
| sparsentan (FILSPARI) | Antagonist | approved | Small molecule | AGTR1 antagonist |
| tasosartan | Antagonist | experimental | Small molecule | AGTR1 antagonist |
| telmisartan (micardis) | Antagonist | approved | Small molecule | AGTR1 antagonist |
| trd205 | Antagonist | experimental | Small molecule | AGTR1 antagonist |
| trv-120027 | Antagonist | experimental | Small molecule | Type-1 angiotensin II receptor antagonist |
| valsartan (diovan) | Antagonist | approved | Small molecule | AGTR1 antagonist |
| cftx-1554 | Inhibitor | experimental | Small molecule | AGTR1 inhibitor |