← Mechanisms of action
ADORA1
SINGLE PROTEINHomo sapiens
Preferred name: Adenosine A1 receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (20)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| amp-579 | Agonist | experimental | Small molecule | ADORA1 agonist |
| bay1067197 | Agonist | experimental | Small molecule | ADORA1 agonist |
| defibrotide (defitelio) | Agonist | approved | Animal product | Adenosine A1 receptor agonist |
| gw493838 | Agonist | experimental | Small molecule | ADORA1 agonist |
| rpr749 | Agonist | experimental | Small molecule | ADORA1 agonist |
| selodenoson | Agonist | experimental | Small molecule | ADORA1 agonist |
| tecadenoson | Agonist | experimental | Small molecule | ADORA1 agonist |
| trabodenoson | Agonist | experimental | Small molecule | ADORA1 agonist |
| derenofylline | Antagonist | experimental | Small molecule | ADORA1 antagonist |
| fk-453 | Antagonist | experimental | Small molecule | ADORA1 antagonist |
| naxifylline | Antagonist | experimental | Small molecule | ADORA1 antagonist |
| pbf-1650 | Antagonist | experimental | Small molecule | ADORA1 antagonist |
| pbf-680 | Antagonist | experimental | Small molecule | ADORA1 antagonist |
| rolofylline | Antagonist | experimental | Small molecule | ADORA1 antagonist |
| tonapofylline | Antagonist | experimental | Small molecule | ADORA1 antagonist |
| t-62 | Inhibitor | experimental | Small molecule | ADORA1 inhibitor |
| t-62 | Modulator | experimental | Small molecule | Adenosine A1 receptor modulator |
| capadenoson | Partial agonist | experimental | Small molecule | ADORA1 partial agonist |
| gs-9667 | Partial agonist | experimental | Small molecule | ADORA1 partial agonist |
| neladenoson bialanate | Partial agonist | experimental | Small molecule | ADORA1 partial agonist |