odiparcil

Small moleculeexperimental

Clinical trial activity

5 trials · 6 clinical orgs · 0 marketing orgs

Phase 1
1
Phase 2
4
Phase 3
0
Phase 4
0

Earliest trial started Jan 1, 2002 (NCT00041509)

Timeline

2000s

  1. Jan 1, 2002

    Earliest Phase 2 Sponsor(trial)

  2. Jan 1, 2006

    Earliest Phase 1 Sponsor(trial)

Indications

Mechanism of action

  • Glycosaminoglycans modulator

    Replaces D-xylose as a substrate of galactosyltransferase I. The resulting β-D-xyloside-bound GAG is soluble and released into the circulation.

  • Unspecified targetUnclear

    unclear

Chemistry & pharmacology

Loading structure…

SMILES

Cc1cc(=O)oc2cc(O[C@@H]3SC[C@@H](O)[C@H](O)[C@H]3O)ccc12
Mol. weight
324.35 g/mol
Lipinski Ro5
Pass
Rule of 3
No
Chirality
Single Stereoisomer
Inorganic
No
Polymer
No

Oral

No

Parenteral

No

Topical

No

Sources

Also known as

  • odiparcil
  • odiparcil
  • odiparcil
  • sb424323
  • sb-424323
  • sb-424323

Clinical trials

NCT IDPhaseStart dateSponsor(s)
NCT03370653Phase 2Dec 13, 2017Centro Hospitalar do Porto, Inventiva Pharma, Johannes Gutenburg University, University of London, University of Lyon
NCT00437242Phase 1Oct 1, 2006GlaxoSmithKline
NCT00240643Phase 2Nov 1, 2005GlaxoSmithKline
NCT00244725Phase 2Sep 1, 2005GlaxoSmithKline
NCT00041509Phase 2Jan 1, 2002GlaxoSmithKline
Showing 5 of 5 trials
Page 1 / 1

Organizations

Research & Development (6)

OrganizationOrg typeTrialsAs lead sponsorPhasesEarliest year
GlaxoSmithKlineFor profit4422002
Centro Hospitalar do PortoAcademic/Hospital1012017
Inventiva PharmaFor profit1112017
Johannes Gutenburg UniversityAcademic/Hospital1012017
University of LondonAcademic/Hospital1012017
University of LyonAcademic/Hospital1012017
6 organizations
Page 1 / 1