mgb-bp-3

Small moleculeexperimental

Clinical trial activity

2 trials · 8 clinical orgs · 0 marketing orgs

Phase 1
1
Phase 2
1
Phase 3
0
Phase 4
0

Earliest trial started Jul 1, 2015 (NCT02518607)

Timeline

2010s

  1. Jan 1, 2015

    Earliest Phase 1 Sponsor(trial)

  2. Jan 1, 2019

    Earliest Phase 2 Sponsor(trial)

Indications

Mechanism of action

  • DNABINDING AGENT

    DNA binding agent

Chemistry & pharmacology

Loading structure…

SMILES

Cn1cc(NC(=O)c2cc(NC(=O)c3ccc(/C=C/c4cnc5ccccc5c4)cc3)cn2C)cc1C(=O)NCCN1CCOCC1
Mol. weight
631.74 g/mol
Lipinski Ro5
1 violation(s)
Rule of 3
No
Chirality
Achiral Molecule
Inorganic
No
Polymer
No

Oral

No

Parenteral

No

Topical

No

Sources

Also known as

  • mgb-bp-3
  • mgb-bp-3
  • mgb-bp-3

Clinical trials

NCT IDPhaseStart dateSponsor(s)
NCT03824795Phase 2Feb 7, 2019MGB Biopharma Limited, Syneos Health
NCT02518607Phase 1Jul 1, 2015Analytical Services International Limited, Cambridge Regulatory Services, Hammersmith Medicines Research, Innovate UK, MGB Biopharma Limited, Synlab Services, Viapath
Showing 2 of 2 trials
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Organizations

Research & Development (8)

OrganizationOrg typeTrialsAs lead sponsorPhasesEarliest year
MGB Biopharma LimitedFor profit2222015
Analytical Services International LimitedFor profit1012015
Cambridge Regulatory ServicesFor profit1012015
Hammersmith Medicines ResearchFor profit1012015
Innovate UKGovernment1012015
Syneos HealthFor profit1012019
Synlab ServicesFor profit1012015
ViapathFor profit1012015
8 organizations
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