iobitridol

Trade name: Xenetix

Small moleculeexperimentalImaging agent

Iobitridol is a pharmaceutical drug used as an iodine-based radiocontrast agent in X-ray imaging. It is injected into blood vessels, joints, or body cavities such as the uterus, and filtered out by the kidneys. Its most common adverse effect is nausea. Severe allergic reactions are rare. — Wikipedia

Clinical trial activity

7 trials · 6 clinical orgs · 0 marketing orgs

Phase 1
1
Phase 2
0
Phase 3
0
Phase 4
5

Earliest trial started May 1, 2006 (NCT00347022)

Timeline

2010s

  1. Jan 1, 2013

    Earliest Phase 1 Sponsor(trial)

Indications

Approved for

Mechanism of action

  • Unspecified targetContrast agent

    contrast agent

Chemistry & pharmacology

Loading structure…

SMILES

CN(CC(O)CO)C(=O)c1c(I)c(NC(=O)C(CO)CO)c(I)c(C(=O)N(C)CC(O)CO)c1I
Mol. weight
835.17 g/mol
Lipinski Ro5
2 violation(s)
Rule of 3
No
Chirality
Racemic Mixture
Inorganic
No
Polymer
No

Oral

No

Parenteral

No

Topical

No

Sources

Also known as

  • 5-(3-hydroxy-2-hydroxymethylpropionamido)-n,n'-dimethyl-n,n'-bis(2,3-dihydroxypropyl)-2,4,6-triiodoisophthalamide
  • iobitridol
  • iobitridol
  • iobitridol
  • iobitridol
  • iobitridol
  • iobitridol
  • iobitridol
  • iobitridol
  • xenetix
  • xenetix
  • xenetix

Clinical trials

NCT IDPhaseStart dateSponsor(s)
NCT04027556N/AJun 27, 2019Seoul National University, Siemens
NCT01908309Early Phase 1 (Phase 1)Apr 1, 2013Azienda Sanitaria Locale 9, Grosseto
NCT01639703Phase 4Apr 30, 2012Guerbet
NCT01255722Phase 4Nov 1, 2010Guerbet, Kantonsspital Lucerne
NCT01254552Phase 4Aug 1, 2010Guerbet, University of Ulsan
NCT00382317Phase 4Aug 1, 2006Guerbet
NCT00347022Phase 4May 1, 2006Guerbet
Showing 7 of 7 trials
Page 1 / 1

Organizations

Research & Development (6)

OrganizationOrg typeTrialsAs lead sponsorPhasesEarliest year
GuerbetFor profit5512006
Azienda Sanitaria Locale 9, GrossetoGovernment1112013
Kantonsspital LucerneAcademic/Hospital1012010
Seoul National UniversityAcademic/Hospital1112019
SiemensFor profit1012019
University of UlsanAcademic/Hospital1012010
6 organizations
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