nsi-189

Small moleculeexperimental

Clinical trial activity

3 trials · 2 clinical orgs · 0 marketing orgs

Phase 1
2
Phase 2
1
Phase 3
0
Phase 4
0

Earliest trial started Feb 1, 2011 (NCT01310881)

Timeline

2010s

  1. Jan 1, 2011

    Earliest Phase 1 Sponsor(trial)

  2. Jan 1, 2016

    Earliest Phase 2 Sponsor(trial)

Indications

Mechanism of action

Chemistry & pharmacology

Loading structure…

SMILES

CC(C)CCNc1ncccc1C(=O)N1CCN(Cc2ccccc2)CC1
Mol. weight
366.51 g/mol
Lipinski Ro5
Pass
Rule of 3
No
Chirality
Achiral Molecule
Inorganic
No
Polymer
No

Oral

No

Parenteral

No

Topical

No

Sources

Also known as

  • nsi-189
  • nsi-189

Clinical trials

NCT IDPhaseStart dateSponsor(s)
NCT02695472Phase 2Mar 1, 2016Seneca Biopharma, Inc.
NCT01520649Phase 1May 1, 2012Seneca Biopharma, Inc.
NCT01310881Phase 1Feb 1, 2011California Clinical Trials, Seneca Biopharma, Inc.
Showing 3 of 3 trials
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Organizations

Research & Development (2)

OrganizationOrg typeTrialsAs lead sponsorPhasesEarliest year
Seneca Biopharma, Inc.For profit3322011
California Clinical TrialsFor profit1012011
2 organizations
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