ap-472
Small moleculeexperimental
Clinical trial activity
0 trials · 0 clinical orgs · 0 marketing orgs
Phase 1
0
Phase 2
0
Phase 3
0
Phase 4
0
Mechanism of action
- Metabotropic glutamate receptorPOSITIVE ALLOSTERIC MODULATOR
Metabotropic glutamate receptor positive allosteric modulator
- Metabotropic glutamate receptor 5 (GRM5) ↗
- Metabotropic glutamate receptor 8 (Grm8) ↗
- Metabotropic glutamate receptor 4 (Grm4) ↗
- Metabotropic glutamate receptor 2 (Grm2) ↗
- Metabotropic glutamate receptor 3 (Grm3) ↗
- Metabotropic glutamate receptor 6 (Grm6) ↗
- Metabotropic glutamate receptor 7 (Grm7) ↗
- Metabotropic glutamate receptor 1 (Grm1) ↗
- Metabotropic glutamate receptor 2
- Metabotropic glutamate receptor 6
- Metabotropic glutamate receptor 8
- Metabotropic glutamate receptor 4
- Metabotropic glutamate receptor 3
- Metabotropic glutamate receptor 5
- Metabotropic glutamate receptor 1
- Metabotropic glutamate receptor 7
- Group II metabotropic glutamate receptor (mGlu2/mGlu3)
Chemistry & pharmacology
Oral
No
Parenteral
No
Topical
No