diphencyprone

Small moleculeexperimental

Diphenylcyclopropenone (diphencyprone) is a topically administered experimental drug intended for treating alopecia areata and alopecia totalis. Topical immunotherapy using diphenylcyclopropenone may also be an effective treatment option for recalcitrant warts. It is not approved by either the Food and Drug Administration or the European Medicines Agency. — Wikipedia

Clinical trial activity

8 trials · 8 clinical orgs · 0 marketing orgs

Phase 1
4
Phase 2
2
Phase 3
1
Phase 4
1

Earliest trial started Oct 1, 2012 (NCT01711684)

Timeline

2010s

  1. Jan 1, 2012

    Earliest Phase 1 Sponsor(trial)

  2. Jan 1, 2015

    Earliest Phase 2 Sponsor(trial)

  3. Jan 1, 2018

    Earliest Phase 3 Sponsor(trial)

Indications

Approved for

Mechanism of action

Chemistry & pharmacology

Loading structure…

SMILES

O=c1c(-c2ccccc2)c1-c1ccccc1
Mol. weight
206.24 g/mol
Lipinski Ro5
Pass
Rule of 3
No
Chirality
Achiral Molecule
Inorganic
No
Polymer
No

Oral

No

Parenteral

No

Topical

No

Sources

Also known as

  • 2,3-diphenyl-2-cyclopropen-1-one
  • diphencyprone
  • diphencyprone
  • diphencyprone
  • diphenylcyclopropenone
  • diphenylcyclopropenone
  • diphenylcyclopropenone
  • diphenylcyclopropenone
  • diphenylcyclopropenone monohydrate
  • dpcp
  • dpcp

Clinical trials

NCT IDPhaseStart dateSponsor(s)
NCT05481658Phase 1Oct 6, 2022Icahn School of Medicine at Mount Sinai
NCT05438290Phase 1Sep 30, 2022Icahn School of Medicine at Mount Sinai
NCT05020496N/AJan 1, 2022University of Alabama, Birmingham
NCT04775979Phase 4Jan 17, 2021Ain Shams University
NCT03651752Phase 3Sep 1, 2018National Alopecia Areata Foundation, University of Minnesota
NCT02640820Phase 2Dec 1, 2015RXi Pharmaceuticals
NCT01978483Phase 1Nov 1, 2013Innovaderm
NCT01711684Phase 1Oct 1, 2012Rockefeller University
Showing 8 of 8 trials
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Organizations

Research & Development (8)

OrganizationOrg typeTrialsAs lead sponsorPhasesEarliest year
Icahn School of Medicine at Mount SinaiAcademic/Hospital2212022
Ain Shams UniversityAcademic/Hospital1112021
InnovadermFor profit1112013
National Alopecia Areata FoundationAcademic/Hospital1012018
Rockefeller UniversityAcademic/Hospital1112012
RXi PharmaceuticalsFor profit1112015
University of Alabama, BirminghamAcademic/Hospital1112022
University of MinnesotaAcademic/Hospital1112018
8 organizations
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